PKRA83 (PKRA7) hydrochloride hydrate is a potent prokineticin (PK2) antagonist, which can compete for the binding of PK2 to its receptors PKR1 and PKR2. PKRA83 hydrochloride hydrate potently inhibits PK2 receptors, with IC50 values of 5.0 nM and 8.2 nM for PKR1 and PKR2, respectively. PKRA83 hydrochloride hydrate has anticancer, anti-arthritis and anti-angiogenic activities. PKRA83 hydrochloride hydrate can penetrate the blood-brain barrier[1][2][3].
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Număr Catalog 804-HY-147056ACategorieAfaceri și industrie > Știință și laboratorFurnizorMedChemExpressGentaurDimensiuneGet quoteTipsingle