PF-06424439 methanesulfonate is an oral, potent and selective imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) inhibitor with an IC50 of 14 nM[1]. PF-06424439 methanesulfonate is slowly reversible, time-dependent inhibitor, which inhibits DGAT2 in a noncompetitive mode with respect to the acyl-CoA substrate[2].
1939.44RON
În stoc
Număr Catalog 804-HY-108341ACategorieAfaceri și industrie > Știință și laboratorFurnizorMedChemExpressGentaurDimensiune10mM/1mLTipsingle